4-1BB Antibodies in Oncology Clinical Trials: A Review

4-1BB is a transmembrane glycoprotein found on T lymphocytes, and signaling through 4-1BB activates and differentiates CD3+ and CD8+ T cells. The ability of 4-1BB to stimulate cytotoxic T-cell responses makes it a promising target for therapeutic cancer immunotherapy development. 4-1BB antibodies ha...

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Main Authors: Robin Schwartz, Keerti Vajrala, Gerald S. Falchook
Format: Article
Language:English
Published: Innovative Healthcare Institute 2025-03-01
Series:Journal of Immunotherapy and Precision Oncology
Subjects:
Online Access:https://jipo.org/doi/pdf/10.36401/JIPO-24-30
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author Robin Schwartz
Keerti Vajrala
Gerald S. Falchook
author_facet Robin Schwartz
Keerti Vajrala
Gerald S. Falchook
author_sort Robin Schwartz
collection DOAJ
description 4-1BB is a transmembrane glycoprotein found on T lymphocytes, and signaling through 4-1BB activates and differentiates CD3+ and CD8+ T cells. The ability of 4-1BB to stimulate cytotoxic T-cell responses makes it a promising target for therapeutic cancer immunotherapy development. 4-1BB antibodies have shown promising antitumor activity in preclinical studies and clinical trials. Common side effects include transaminase elevation, cytopenias, fatigue, and nausea. This clinical review summarizes past and current 4-1BB antibodies in oncology clinical trials.
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issn 2666-2345
2590-017X
language English
publishDate 2025-03-01
publisher Innovative Healthcare Institute
record_format Article
series Journal of Immunotherapy and Precision Oncology
spelling doaj-art-1e202b1fda6e4642802b04bc0bdd1c492025-08-20T02:03:07ZengInnovative Healthcare InstituteJournal of Immunotherapy and Precision Oncology2666-23452590-017X2025-03-018212113110.36401/JIPO-24-30i2590-017X-8-2-1214-1BB Antibodies in Oncology Clinical Trials: A ReviewRobin Schwartz0Keerti Vajrala1Gerald S. Falchook2https://orcid.org/0000-0001-9165-21911 Sarah Cannon Research Institute at HealthONE, Denver, CO, USA2 Kansas City University College of Osteopathic Medicine, Kansas City, MO, USA1 Sarah Cannon Research Institute at HealthONE, Denver, CO, USA4-1BB is a transmembrane glycoprotein found on T lymphocytes, and signaling through 4-1BB activates and differentiates CD3+ and CD8+ T cells. The ability of 4-1BB to stimulate cytotoxic T-cell responses makes it a promising target for therapeutic cancer immunotherapy development. 4-1BB antibodies have shown promising antitumor activity in preclinical studies and clinical trials. Common side effects include transaminase elevation, cytopenias, fatigue, and nausea. This clinical review summarizes past and current 4-1BB antibodies in oncology clinical trials.https://jipo.org/doi/pdf/10.36401/JIPO-24-304-1bbcd137clinical trialimmunotherapy
spellingShingle Robin Schwartz
Keerti Vajrala
Gerald S. Falchook
4-1BB Antibodies in Oncology Clinical Trials: A Review
Journal of Immunotherapy and Precision Oncology
4-1bb
cd137
clinical trial
immunotherapy
title 4-1BB Antibodies in Oncology Clinical Trials: A Review
title_full 4-1BB Antibodies in Oncology Clinical Trials: A Review
title_fullStr 4-1BB Antibodies in Oncology Clinical Trials: A Review
title_full_unstemmed 4-1BB Antibodies in Oncology Clinical Trials: A Review
title_short 4-1BB Antibodies in Oncology Clinical Trials: A Review
title_sort 4 1bb antibodies in oncology clinical trials a review
topic 4-1bb
cd137
clinical trial
immunotherapy
url https://jipo.org/doi/pdf/10.36401/JIPO-24-30
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AT keertivajrala 41bbantibodiesinoncologyclinicaltrialsareview
AT geraldsfalchook 41bbantibodiesinoncologyclinicaltrialsareview