COMPARATIVE STUDY OF INTERACTION OF SOME DOMESTIC HUMAN INSULIN SUBSTANCES AND ITS ANALOGUES WITH INSULIN RECEPTOR BY METHOD OF SURFACE PLASMON RESONANCE

The high demand for insulin preparations by the population of the country makes it urgent to create domestic bioanalogues for the treatment of diabetes mellitus. The equivalency of the quality, safety and efficacy of the bioanalogue with the reference medicinal preparation registered in Russia is re...

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Main Authors: I. N. Urakova, K. L. Kryshen, O. N. Pozharitskaya, M. V. Gavrilin, A. N. Shikov, M. N. Makarova, V. G. Makarov
Format: Article
Language:Russian
Published: LLC Center of Pharmaceutical Analytics (LLC «CPHA») 2019-01-01
Series:Разработка и регистрация лекарственных средств
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Online Access:https://www.pharmjournal.ru/jour/article/view/616
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author I. N. Urakova
K. L. Kryshen
O. N. Pozharitskaya
M. V. Gavrilin
A. N. Shikov
M. N. Makarova
V. G. Makarov
author_facet I. N. Urakova
K. L. Kryshen
O. N. Pozharitskaya
M. V. Gavrilin
A. N. Shikov
M. N. Makarova
V. G. Makarov
author_sort I. N. Urakova
collection DOAJ
description The high demand for insulin preparations by the population of the country makes it urgent to create domestic bioanalogues for the treatment of diabetes mellitus. The equivalency of the quality, safety and efficacy of the bioanalogue with the reference medicinal preparation registered in Russia is required by authority at the stage of preclinical studies. The aim of the study was to study the interaction of insulin substances of domestic production, including short and long-acting insulin with the insulin receptor in comparison with the reference substances registered in Russia by the surface plasmon resonance method. Comparing the interaction kinetics curves and calculated dissociation constants determined by the surface plasmon resonance method it was confirmed that there are no statistically significant differences between the potentially bioanalogical insulin substances Rosinsulin R, Rosinsulin Glargin and Rosinsulin Aspart (LLC ”Zavod Medsintez”, Russia) and the corresponding substances of registered in Russia medicines.
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institution DOAJ
issn 2305-2066
2658-5049
language Russian
publishDate 2019-01-01
publisher LLC Center of Pharmaceutical Analytics (LLC «CPHA»)
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series Разработка и регистрация лекарственных средств
spelling doaj-art-1ce592b7cc1249b699ea5e3caac3a0b92025-08-20T02:54:18ZrusLLC Center of Pharmaceutical Analytics (LLC «CPHA»)Разработка и регистрация лекарственных средств2305-20662658-50492019-01-0103136143616COMPARATIVE STUDY OF INTERACTION OF SOME DOMESTIC HUMAN INSULIN SUBSTANCES AND ITS ANALOGUES WITH INSULIN RECEPTOR BY METHOD OF SURFACE PLASMON RESONANCEI. N. Urakova0K. L. Kryshen1O. N. Pozharitskaya2M. V. Gavrilin3A. N. Shikov4M. N. Makarova5V. G. Makarov6St.-Petersburg Institute of PharmacyRMC «HOUSE OF PHARMACY» JSCSt.-Petersburg Institute of PharmacyLLC «Zavod Medsintez»St.-Petersburg Institute of PharmacyRMC «HOUSE OF PHARMACY» JSCRMC «HOUSE OF PHARMACY» JSCThe high demand for insulin preparations by the population of the country makes it urgent to create domestic bioanalogues for the treatment of diabetes mellitus. The equivalency of the quality, safety and efficacy of the bioanalogue with the reference medicinal preparation registered in Russia is required by authority at the stage of preclinical studies. The aim of the study was to study the interaction of insulin substances of domestic production, including short and long-acting insulin with the insulin receptor in comparison with the reference substances registered in Russia by the surface plasmon resonance method. Comparing the interaction kinetics curves and calculated dissociation constants determined by the surface plasmon resonance method it was confirmed that there are no statistically significant differences between the potentially bioanalogical insulin substances Rosinsulin R, Rosinsulin Glargin and Rosinsulin Aspart (LLC ”Zavod Medsintez”, Russia) and the corresponding substances of registered in Russia medicines.https://www.pharmjournal.ru/jour/article/view/616inslulininslulin glargininsulin aspartinsulin receptorsplasmon resonanceassociation constant
spellingShingle I. N. Urakova
K. L. Kryshen
O. N. Pozharitskaya
M. V. Gavrilin
A. N. Shikov
M. N. Makarova
V. G. Makarov
COMPARATIVE STUDY OF INTERACTION OF SOME DOMESTIC HUMAN INSULIN SUBSTANCES AND ITS ANALOGUES WITH INSULIN RECEPTOR BY METHOD OF SURFACE PLASMON RESONANCE
Разработка и регистрация лекарственных средств
inslulin
inslulin glargin
insulin aspart
insulin receptors
plasmon resonance
association constant
title COMPARATIVE STUDY OF INTERACTION OF SOME DOMESTIC HUMAN INSULIN SUBSTANCES AND ITS ANALOGUES WITH INSULIN RECEPTOR BY METHOD OF SURFACE PLASMON RESONANCE
title_full COMPARATIVE STUDY OF INTERACTION OF SOME DOMESTIC HUMAN INSULIN SUBSTANCES AND ITS ANALOGUES WITH INSULIN RECEPTOR BY METHOD OF SURFACE PLASMON RESONANCE
title_fullStr COMPARATIVE STUDY OF INTERACTION OF SOME DOMESTIC HUMAN INSULIN SUBSTANCES AND ITS ANALOGUES WITH INSULIN RECEPTOR BY METHOD OF SURFACE PLASMON RESONANCE
title_full_unstemmed COMPARATIVE STUDY OF INTERACTION OF SOME DOMESTIC HUMAN INSULIN SUBSTANCES AND ITS ANALOGUES WITH INSULIN RECEPTOR BY METHOD OF SURFACE PLASMON RESONANCE
title_short COMPARATIVE STUDY OF INTERACTION OF SOME DOMESTIC HUMAN INSULIN SUBSTANCES AND ITS ANALOGUES WITH INSULIN RECEPTOR BY METHOD OF SURFACE PLASMON RESONANCE
title_sort comparative study of interaction of some domestic human insulin substances and its analogues with insulin receptor by method of surface plasmon resonance
topic inslulin
inslulin glargin
insulin aspart
insulin receptors
plasmon resonance
association constant
url https://www.pharmjournal.ru/jour/article/view/616
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