Microbial Fermentation Affects the Structure–Activity Relationship of Bioactive Compounds in Ginseng and Its Applications in Fermentation Products: A Review

Microbial fermentation technology has emerged as a pivotal approach for enhancing ginseng efficacy through the transformation of active ingredient molecular structures. This paper reviews the impact of microbial fermentation on the structure–activity relationship of ginseng bioactive compounds and a...

Full description

Saved in:
Bibliographic Details
Main Authors: Juan Bai, Zixian Zhu, Wei Luo, Miran Jang, Beibei Pan, Ying Zhu, Jiayan Zhang, Yansheng Zhao, Xiang Xiao
Format: Article
Language:English
Published: MDPI AG 2025-07-01
Series:Foods
Subjects:
Online Access:https://www.mdpi.com/2304-8158/14/14/2473
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1849409537536163840
author Juan Bai
Zixian Zhu
Wei Luo
Miran Jang
Beibei Pan
Ying Zhu
Jiayan Zhang
Yansheng Zhao
Xiang Xiao
author_facet Juan Bai
Zixian Zhu
Wei Luo
Miran Jang
Beibei Pan
Ying Zhu
Jiayan Zhang
Yansheng Zhao
Xiang Xiao
author_sort Juan Bai
collection DOAJ
description Microbial fermentation technology has emerged as a pivotal approach for enhancing ginseng efficacy through the transformation of active ingredient molecular structures. This paper reviews the impact of microbial fermentation on the structure–activity relationship of ginseng bioactive compounds and advances in its application. Bibliometric analysis indicates that <i>Panax</i> species (<i>Panax ginseng</i>, <i>Panax notoginseng</i>) are primarily fermented using lactic acid bacteria and <i>Aspergillus</i> spp., with research predominantly focused on conversion efficiency to rare ginsenosides (Compound K, Rg3, and Rh2). Specifically, this review details the biotransformation pathways of these rare ginsenosides and the resultant bioactivity enhancements. Additionally, it summarizes the effects of other microorganisms, such as fungal fruiting bodies, on additional ginseng constituents like polysaccharides and polyphenols. Microbial fermentation has been successfully implemented in functional products, including ginseng vinegar, wine, and fermented milk. This review subsequently examines these applications, emphasizing fermentation’s potential to enhance product functionality. However, challenges remain in strain screening, process standardization, and analysis of multi-component synergistic mechanisms. In summary, this review synthesizes recent advancements in understanding the mechanisms of microbial fermentation on ginseng and its translational applications in functional foods and pharmaceuticals.
format Article
id doaj-art-183b0cc8e3a14f619f679979735eaae2
institution Kabale University
issn 2304-8158
language English
publishDate 2025-07-01
publisher MDPI AG
record_format Article
series Foods
spelling doaj-art-183b0cc8e3a14f619f679979735eaae22025-08-20T03:35:28ZengMDPI AGFoods2304-81582025-07-011414247310.3390/foods14142473Microbial Fermentation Affects the Structure–Activity Relationship of Bioactive Compounds in Ginseng and Its Applications in Fermentation Products: A ReviewJuan Bai0Zixian Zhu1Wei Luo2Miran Jang3Beibei Pan4Ying Zhu5Jiayan Zhang6Yansheng Zhao7Xiang Xiao8School of Food and Biological Engineering, Jiangsu University, Zhenjiang 212013, ChinaSchool of Food and Biological Engineering, Jiangsu University, Zhenjiang 212013, ChinaSchool of Food and Biological Engineering, Jiangsu University, Zhenjiang 212013, ChinaDepartment of Institute of Digital Anti-Aging Healthcare, Inje University, Gimhae 50834, Republic of KoreaSchool of Food and Biological Engineering, Jiangsu University, Zhenjiang 212013, ChinaSchool of Food and Biological Engineering, Jiangsu University, Zhenjiang 212013, ChinaSchool of Food and Biological Engineering, Jiangsu University, Zhenjiang 212013, ChinaSchool of Food and Biological Engineering, Jiangsu University, Zhenjiang 212013, ChinaSchool of Food and Biological Engineering, Jiangsu University, Zhenjiang 212013, ChinaMicrobial fermentation technology has emerged as a pivotal approach for enhancing ginseng efficacy through the transformation of active ingredient molecular structures. This paper reviews the impact of microbial fermentation on the structure–activity relationship of ginseng bioactive compounds and advances in its application. Bibliometric analysis indicates that <i>Panax</i> species (<i>Panax ginseng</i>, <i>Panax notoginseng</i>) are primarily fermented using lactic acid bacteria and <i>Aspergillus</i> spp., with research predominantly focused on conversion efficiency to rare ginsenosides (Compound K, Rg3, and Rh2). Specifically, this review details the biotransformation pathways of these rare ginsenosides and the resultant bioactivity enhancements. Additionally, it summarizes the effects of other microorganisms, such as fungal fruiting bodies, on additional ginseng constituents like polysaccharides and polyphenols. Microbial fermentation has been successfully implemented in functional products, including ginseng vinegar, wine, and fermented milk. This review subsequently examines these applications, emphasizing fermentation’s potential to enhance product functionality. However, challenges remain in strain screening, process standardization, and analysis of multi-component synergistic mechanisms. In summary, this review synthesizes recent advancements in understanding the mechanisms of microbial fermentation on ginseng and its translational applications in functional foods and pharmaceuticals.https://www.mdpi.com/2304-8158/14/14/2473biotransformationfermentationfermented productsginsengstructure–activity relationship
spellingShingle Juan Bai
Zixian Zhu
Wei Luo
Miran Jang
Beibei Pan
Ying Zhu
Jiayan Zhang
Yansheng Zhao
Xiang Xiao
Microbial Fermentation Affects the Structure–Activity Relationship of Bioactive Compounds in Ginseng and Its Applications in Fermentation Products: A Review
Foods
biotransformation
fermentation
fermented products
ginseng
structure–activity relationship
title Microbial Fermentation Affects the Structure–Activity Relationship of Bioactive Compounds in Ginseng and Its Applications in Fermentation Products: A Review
title_full Microbial Fermentation Affects the Structure–Activity Relationship of Bioactive Compounds in Ginseng and Its Applications in Fermentation Products: A Review
title_fullStr Microbial Fermentation Affects the Structure–Activity Relationship of Bioactive Compounds in Ginseng and Its Applications in Fermentation Products: A Review
title_full_unstemmed Microbial Fermentation Affects the Structure–Activity Relationship of Bioactive Compounds in Ginseng and Its Applications in Fermentation Products: A Review
title_short Microbial Fermentation Affects the Structure–Activity Relationship of Bioactive Compounds in Ginseng and Its Applications in Fermentation Products: A Review
title_sort microbial fermentation affects the structure activity relationship of bioactive compounds in ginseng and its applications in fermentation products a review
topic biotransformation
fermentation
fermented products
ginseng
structure–activity relationship
url https://www.mdpi.com/2304-8158/14/14/2473
work_keys_str_mv AT juanbai microbialfermentationaffectsthestructureactivityrelationshipofbioactivecompoundsinginsenganditsapplicationsinfermentationproductsareview
AT zixianzhu microbialfermentationaffectsthestructureactivityrelationshipofbioactivecompoundsinginsenganditsapplicationsinfermentationproductsareview
AT weiluo microbialfermentationaffectsthestructureactivityrelationshipofbioactivecompoundsinginsenganditsapplicationsinfermentationproductsareview
AT miranjang microbialfermentationaffectsthestructureactivityrelationshipofbioactivecompoundsinginsenganditsapplicationsinfermentationproductsareview
AT beibeipan microbialfermentationaffectsthestructureactivityrelationshipofbioactivecompoundsinginsenganditsapplicationsinfermentationproductsareview
AT yingzhu microbialfermentationaffectsthestructureactivityrelationshipofbioactivecompoundsinginsenganditsapplicationsinfermentationproductsareview
AT jiayanzhang microbialfermentationaffectsthestructureactivityrelationshipofbioactivecompoundsinginsenganditsapplicationsinfermentationproductsareview
AT yanshengzhao microbialfermentationaffectsthestructureactivityrelationshipofbioactivecompoundsinginsenganditsapplicationsinfermentationproductsareview
AT xiangxiao microbialfermentationaffectsthestructureactivityrelationshipofbioactivecompoundsinginsenganditsapplicationsinfermentationproductsareview