Targeting CD38 in Antibody-Mediated Rejection

Antibody-mediated rejection (AMR) remains a major challenge in clinical transplantation. Current therapies have yielded inconsistent outcomes, highlighting the need for innovative approaches. CD38, a multifunctional glycoprotein, is highly expressed on plasma cells and natural killer (NK) cells, pot...

Full description

Saved in:
Bibliographic Details
Main Authors: Katharina A. Mayer, Klemens Budde, Matthias Diebold, Philip F. Halloran, Georg A. Böhmig
Format: Article
Language:English
Published: Frontiers Media S.A. 2025-05-01
Series:Transplant International
Subjects:
Online Access:https://www.frontierspartnerships.org/articles/10.3389/ti.2025.14343/full
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1849727147423301632
author Katharina A. Mayer
Klemens Budde
Matthias Diebold
Matthias Diebold
Philip F. Halloran
Georg A. Böhmig
author_facet Katharina A. Mayer
Klemens Budde
Matthias Diebold
Matthias Diebold
Philip F. Halloran
Georg A. Böhmig
author_sort Katharina A. Mayer
collection DOAJ
description Antibody-mediated rejection (AMR) remains a major challenge in clinical transplantation. Current therapies have yielded inconsistent outcomes, highlighting the need for innovative approaches. CD38, a multifunctional glycoprotein, is highly expressed on plasma cells and natural killer (NK) cells, potentially offering a dual mechanism of action that could intervene in the pathophysiologic course of AMR: depleting alloantibody-producing plasma cells and NK cells. This review focuses on recent results from CD38-targeted therapies, with felzartamab emerging as a promising option. Previous case reports and series suggested that off-label daratumumab treatment could effectively reverse AMR. Felzartamab has now demonstrated safety and efficacy in a phase 2 trial for late AMR. Reductions in microvascular inflammation, downregulation of rejection-associated transcripts, and decreases in donor-derived cell-free DNA paralleled a substantial decrease in NK cell counts. However, felzartamab did not significantly affect donor-specific antibodies, which may reflect its distinct mechanism of action, primarily involving antibody-dependent cellular cytotoxicity and phagocytosis. The effects on rejection activity may have a rapid onset, but are transient. The potential benefits of prolonged therapy are currently being investigated in a recently launched phase III trial. Future studies may expand the applications of CD38 targeting to early AMR or broader indications, such as DSA-negative microvascular inflammation.
format Article
id doaj-art-13e091aa21d04084a3e41cfaaf1e4ea6
institution DOAJ
issn 1432-2277
language English
publishDate 2025-05-01
publisher Frontiers Media S.A.
record_format Article
series Transplant International
spelling doaj-art-13e091aa21d04084a3e41cfaaf1e4ea62025-08-20T03:09:57ZengFrontiers Media S.A.Transplant International1432-22772025-05-013810.3389/ti.2025.1434314343Targeting CD38 in Antibody-Mediated RejectionKatharina A. Mayer0Klemens Budde1Matthias Diebold2Matthias Diebold3Philip F. Halloran4Georg A. Böhmig5Division of Nephrology and Dialysis, Department of Medicine III, Medical University of Vienna, Vienna, AustriaDepartment of Nephrology, Charité Universitätsmedizin Berlin, Berlin, GermanyDivision of Nephrology and Dialysis, Department of Medicine III, Medical University of Vienna, Vienna, AustriaClinic for Transplantation Immunology and Nephrology, University Hospital Basel, University of Basel, Basel, SwitzerlandAlberta Transplant Applied Genomics Centre, Faculty of Medicine and Dentistry, University of Alberta, Edmonton, AB, CanadaDivision of Nephrology and Dialysis, Department of Medicine III, Medical University of Vienna, Vienna, AustriaAntibody-mediated rejection (AMR) remains a major challenge in clinical transplantation. Current therapies have yielded inconsistent outcomes, highlighting the need for innovative approaches. CD38, a multifunctional glycoprotein, is highly expressed on plasma cells and natural killer (NK) cells, potentially offering a dual mechanism of action that could intervene in the pathophysiologic course of AMR: depleting alloantibody-producing plasma cells and NK cells. This review focuses on recent results from CD38-targeted therapies, with felzartamab emerging as a promising option. Previous case reports and series suggested that off-label daratumumab treatment could effectively reverse AMR. Felzartamab has now demonstrated safety and efficacy in a phase 2 trial for late AMR. Reductions in microvascular inflammation, downregulation of rejection-associated transcripts, and decreases in donor-derived cell-free DNA paralleled a substantial decrease in NK cell counts. However, felzartamab did not significantly affect donor-specific antibodies, which may reflect its distinct mechanism of action, primarily involving antibody-dependent cellular cytotoxicity and phagocytosis. The effects on rejection activity may have a rapid onset, but are transient. The potential benefits of prolonged therapy are currently being investigated in a recently launched phase III trial. Future studies may expand the applications of CD38 targeting to early AMR or broader indications, such as DSA-negative microvascular inflammation.https://www.frontierspartnerships.org/articles/10.3389/ti.2025.14343/fullantibody-mediated rejectionCD38natural killer cellskidney transplantationtreatment
spellingShingle Katharina A. Mayer
Klemens Budde
Matthias Diebold
Matthias Diebold
Philip F. Halloran
Georg A. Böhmig
Targeting CD38 in Antibody-Mediated Rejection
Transplant International
antibody-mediated rejection
CD38
natural killer cells
kidney transplantation
treatment
title Targeting CD38 in Antibody-Mediated Rejection
title_full Targeting CD38 in Antibody-Mediated Rejection
title_fullStr Targeting CD38 in Antibody-Mediated Rejection
title_full_unstemmed Targeting CD38 in Antibody-Mediated Rejection
title_short Targeting CD38 in Antibody-Mediated Rejection
title_sort targeting cd38 in antibody mediated rejection
topic antibody-mediated rejection
CD38
natural killer cells
kidney transplantation
treatment
url https://www.frontierspartnerships.org/articles/10.3389/ti.2025.14343/full
work_keys_str_mv AT katharinaamayer targetingcd38inantibodymediatedrejection
AT klemensbudde targetingcd38inantibodymediatedrejection
AT matthiasdiebold targetingcd38inantibodymediatedrejection
AT matthiasdiebold targetingcd38inantibodymediatedrejection
AT philipfhalloran targetingcd38inantibodymediatedrejection
AT georgabohmig targetingcd38inantibodymediatedrejection