Gold Nanorods Targeted to Delta Opioid Receptor: Plasmon-Resonant Contrast and Photothermal Agents

Molecularly targeted gold nanorods were investigated for applications in both diagnostic imaging and disease treatment with cellular resolution. The nanorods were tested in two genetically engineered cell lines derived from the human colon carcinoma HCT-116, a model for studying ligand-receptor inte...

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Main Authors: Kvar C. Black, Nathaniel D. Kirkpatrick, Timothy S. Troutman, Liping Xu, Josef Vagner, Robert J. Gillies, Jennifer K. Barton, Urs Utzinger, Marek Romanowski
Format: Article
Language:English
Published: SAGE Publishing 2008-01-01
Series:Molecular Imaging
Online Access:https://doi.org/10.2310/7290.2008.0007
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author Kvar C. Black
Nathaniel D. Kirkpatrick
Timothy S. Troutman
Liping Xu
Josef Vagner
Robert J. Gillies
Jennifer K. Barton
Urs Utzinger
Marek Romanowski
author_facet Kvar C. Black
Nathaniel D. Kirkpatrick
Timothy S. Troutman
Liping Xu
Josef Vagner
Robert J. Gillies
Jennifer K. Barton
Urs Utzinger
Marek Romanowski
author_sort Kvar C. Black
collection DOAJ
description Molecularly targeted gold nanorods were investigated for applications in both diagnostic imaging and disease treatment with cellular resolution. The nanorods were tested in two genetically engineered cell lines derived from the human colon carcinoma HCT-116, a model for studying ligand-receptor interactions. One of these lines was modified to express delta opioid receptor (δOR) and green fluorescent protein, whereas the other was receptor free and expressed a red fluorescent protein, to serve as the control. Deltorphin, a high-affinity ligand for δOR, was stably attached to the gold nanorods through a thiol-terminated linker. In a mixed population of cells, we demonstrated selective imaging and destruction of receptor-expressing cells while sparing those cells that did not express the receptor. The molecularly targeted nanorods can be used as an in vitro ligand-binding and cytotoxic treatment assay platform and could potentially be applied in vivo for diagnostic and therapeutic purposes with endoscopic technology.
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spelling doaj-art-12eadd0bcd9a4cec8b9a479025cf16032025-08-20T02:43:13ZengSAGE PublishingMolecular Imaging1536-01212008-01-01710.2310/7290.2008.000710.2310_7290.2008.0007Gold Nanorods Targeted to Delta Opioid Receptor: Plasmon-Resonant Contrast and Photothermal AgentsKvar C. BlackNathaniel D. KirkpatrickTimothy S. TroutmanLiping XuJosef VagnerRobert J. GilliesJennifer K. BartonUrs UtzingerMarek RomanowskiMolecularly targeted gold nanorods were investigated for applications in both diagnostic imaging and disease treatment with cellular resolution. The nanorods were tested in two genetically engineered cell lines derived from the human colon carcinoma HCT-116, a model for studying ligand-receptor interactions. One of these lines was modified to express delta opioid receptor (δOR) and green fluorescent protein, whereas the other was receptor free and expressed a red fluorescent protein, to serve as the control. Deltorphin, a high-affinity ligand for δOR, was stably attached to the gold nanorods through a thiol-terminated linker. In a mixed population of cells, we demonstrated selective imaging and destruction of receptor-expressing cells while sparing those cells that did not express the receptor. The molecularly targeted nanorods can be used as an in vitro ligand-binding and cytotoxic treatment assay platform and could potentially be applied in vivo for diagnostic and therapeutic purposes with endoscopic technology.https://doi.org/10.2310/7290.2008.0007
spellingShingle Kvar C. Black
Nathaniel D. Kirkpatrick
Timothy S. Troutman
Liping Xu
Josef Vagner
Robert J. Gillies
Jennifer K. Barton
Urs Utzinger
Marek Romanowski
Gold Nanorods Targeted to Delta Opioid Receptor: Plasmon-Resonant Contrast and Photothermal Agents
Molecular Imaging
title Gold Nanorods Targeted to Delta Opioid Receptor: Plasmon-Resonant Contrast and Photothermal Agents
title_full Gold Nanorods Targeted to Delta Opioid Receptor: Plasmon-Resonant Contrast and Photothermal Agents
title_fullStr Gold Nanorods Targeted to Delta Opioid Receptor: Plasmon-Resonant Contrast and Photothermal Agents
title_full_unstemmed Gold Nanorods Targeted to Delta Opioid Receptor: Plasmon-Resonant Contrast and Photothermal Agents
title_short Gold Nanorods Targeted to Delta Opioid Receptor: Plasmon-Resonant Contrast and Photothermal Agents
title_sort gold nanorods targeted to delta opioid receptor plasmon resonant contrast and photothermal agents
url https://doi.org/10.2310/7290.2008.0007
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