Vitamin D Receptor Agonists Target CXCL10: New Therapeutic Tools for Resolution of Inflammation

Understanding the many biological extraskeletal actions of vitamin D has increased in the past decades. Indeed, vitamin D and analogue molecules, besides the classical actions on bone metabolism, exert several beneficial effects on metabolic homeostasis, heart-cardiovascular, brain, and muscle physi...

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Main Authors: Sabino Scolletta, Marta Colletti, Luigi Di Luigi, Clara Crescioli
Format: Article
Language:English
Published: Wiley 2013-01-01
Series:Mediators of Inflammation
Online Access:http://dx.doi.org/10.1155/2013/876319
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author Sabino Scolletta
Marta Colletti
Luigi Di Luigi
Clara Crescioli
author_facet Sabino Scolletta
Marta Colletti
Luigi Di Luigi
Clara Crescioli
author_sort Sabino Scolletta
collection DOAJ
description Understanding the many biological extraskeletal actions of vitamin D has increased in the past decades. Indeed, vitamin D and analogue molecules, besides the classical actions on bone metabolism, exert several beneficial effects on metabolic homeostasis, heart-cardiovascular, brain, and muscle physiological functions, throughout the interaction with the specific vitamin D receptor (VDR). In particular, VDR agonists powerfully control innate and adaptive immune system with favorable effects on human health. VDR ligands act as immunomodulators that are potent enough to retain anti-inflammatory effects, even though the mechanism underlying those effects is not yet fully elucidated. VDR agonists exert a significant suppression of inflammatory processes switching the immune response from T helper 1 (Th1) to T helper 2 (Th2) dominance and counteracting the self-enhancing inflammatory loop between immune and resident cells, especially by cytokine release impairment. Those molecules are able, indeed, to reduce the release of the interferon (IFN)-induced 10 kDa protein IP-10/CXCL10, a powerful chemokine driving Th1-mediated inflammation. Based on their features, VDR ligands show the potentiality to be included in immunosuppressive regimens, aimed to control auto- and alloimmune Th1-driven overreactivity, occurring, for example, in autoimmune disease or graft rejection.
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issn 0962-9351
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language English
publishDate 2013-01-01
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series Mediators of Inflammation
spelling doaj-art-10fde73026ba4f2d9732c0980f805b522025-08-20T03:55:45ZengWileyMediators of Inflammation0962-93511466-18612013-01-01201310.1155/2013/876319876319Vitamin D Receptor Agonists Target CXCL10: New Therapeutic Tools for Resolution of InflammationSabino Scolletta0Marta Colletti1Luigi Di Luigi2Clara Crescioli3Department of Medical Biotechnologies, University of Siena, Viale Bracci 1, 53100 Siena, ItalyDepartment of Movement, Human and Health Sciences, Unit of Endocrinology, University of Rome Foro Italico, Piazza Lauro de Bosis 15, 00135 Rome, ItalyDepartment of Movement, Human and Health Sciences, Unit of Endocrinology, University of Rome Foro Italico, Piazza Lauro de Bosis 15, 00135 Rome, ItalyDepartment of Movement, Human and Health Sciences, Unit of Endocrinology, University of Rome Foro Italico, Piazza Lauro de Bosis 15, 00135 Rome, ItalyUnderstanding the many biological extraskeletal actions of vitamin D has increased in the past decades. Indeed, vitamin D and analogue molecules, besides the classical actions on bone metabolism, exert several beneficial effects on metabolic homeostasis, heart-cardiovascular, brain, and muscle physiological functions, throughout the interaction with the specific vitamin D receptor (VDR). In particular, VDR agonists powerfully control innate and adaptive immune system with favorable effects on human health. VDR ligands act as immunomodulators that are potent enough to retain anti-inflammatory effects, even though the mechanism underlying those effects is not yet fully elucidated. VDR agonists exert a significant suppression of inflammatory processes switching the immune response from T helper 1 (Th1) to T helper 2 (Th2) dominance and counteracting the self-enhancing inflammatory loop between immune and resident cells, especially by cytokine release impairment. Those molecules are able, indeed, to reduce the release of the interferon (IFN)-induced 10 kDa protein IP-10/CXCL10, a powerful chemokine driving Th1-mediated inflammation. Based on their features, VDR ligands show the potentiality to be included in immunosuppressive regimens, aimed to control auto- and alloimmune Th1-driven overreactivity, occurring, for example, in autoimmune disease or graft rejection.http://dx.doi.org/10.1155/2013/876319
spellingShingle Sabino Scolletta
Marta Colletti
Luigi Di Luigi
Clara Crescioli
Vitamin D Receptor Agonists Target CXCL10: New Therapeutic Tools for Resolution of Inflammation
Mediators of Inflammation
title Vitamin D Receptor Agonists Target CXCL10: New Therapeutic Tools for Resolution of Inflammation
title_full Vitamin D Receptor Agonists Target CXCL10: New Therapeutic Tools for Resolution of Inflammation
title_fullStr Vitamin D Receptor Agonists Target CXCL10: New Therapeutic Tools for Resolution of Inflammation
title_full_unstemmed Vitamin D Receptor Agonists Target CXCL10: New Therapeutic Tools for Resolution of Inflammation
title_short Vitamin D Receptor Agonists Target CXCL10: New Therapeutic Tools for Resolution of Inflammation
title_sort vitamin d receptor agonists target cxcl10 new therapeutic tools for resolution of inflammation
url http://dx.doi.org/10.1155/2013/876319
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