Acoustic ejection mass spectrometry: An integrated pipeline for ultra-high throughput screening, reactivity profiling, and potency analysis of covalent BTK inhibitors

Covalent drug discovery has garnered renewed interest due to its potential to target proteins previously considered ''undruggable.'' Intact protein mass spectrometry (MS) is a critical technique for providing direct evidence of covalent drug modifications to protein targets. Howe...

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Bibliographic Details
Main Authors: Ronghai Cheng, Adil Muneer, Maria Hercher, Bekim Bajrami, Reza Nemati
Format: Article
Language:English
Published: Elsevier 2025-08-01
Series:SLAS Technology
Subjects:
Online Access:http://www.sciencedirect.com/science/article/pii/S2472630325000652
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