Bioassay-guided isolation of anti-hepatitis B virus flavonoid myricetin-3-O-rhamnoside along with quercetin from Guiera senegalensis leaves

Recently, we have shown in vitro anti-hepatitis B virus (HBV) activity of G. senegalensis J.F. Gmel leaves, and Identified quercetin and other flavonoids by HPTLC. Here we report bioassay-directed fractionation of G. senegalensis leaves using column chromatography and isolation of two flavonoinds fr...

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Main Authors: Mohammad K. Parvez, Mohammed S. Al-Dosari, Ahmed H. Arbab, Adnan J. Al-Rehaily, Mazin A.S. Abdelwahid
Format: Article
Language:English
Published: Springer 2020-05-01
Series:Saudi Pharmaceutical Journal
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Online Access:http://www.sciencedirect.com/science/article/pii/S131901642030061X
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author Mohammad K. Parvez
Mohammed S. Al-Dosari
Ahmed H. Arbab
Adnan J. Al-Rehaily
Mazin A.S. Abdelwahid
author_facet Mohammad K. Parvez
Mohammed S. Al-Dosari
Ahmed H. Arbab
Adnan J. Al-Rehaily
Mazin A.S. Abdelwahid
author_sort Mohammad K. Parvez
collection DOAJ
description Recently, we have shown in vitro anti-hepatitis B virus (HBV) activity of G. senegalensis J.F. Gmel leaves, and Identified quercetin and other flavonoids by HPTLC. Here we report bioassay-directed fractionation of G. senegalensis leaves using column chromatography and isolation of two flavonoinds from the n-butanol fraction, their structure determination (1H NMR, 13C NMR and 2D-NMR) and assessment of antiviral activities (HBsAg and HBeAg assay) in HBV-reporter HepG2.2.2.15 cells. Further molecular docking was performed against HBV polymerase (Pol/RT) and capsid (Core) proteins as well as host-receptor sodium taurocholate co-transporting polypeptide (NTCP). The two isolated bioactive compounds were identified as quercetin and myricetin-3-O-rhamnoside. Quercetin significantly inhibited synthesis of HBsAg and HBeAg by about 60% and 62%, respectively as compared to myricetin-3-O-rhamnoside by 44% and 35%, respectively. Molecular docking of the two anti-HBV flavonoids revealed their higher binding affinities towards Pol/RT than Core and NTCP. In conclusion, this is the first report on anti-HBV active myricetin-3-O-rhamnoside along with quercetin isolated from G. senegalensis leaves. Their possible mode of anti-HBV activities are suggested through binding with viral Pol/RT and Core as well as host NTCP proteins.
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spelling doaj-art-06e2ec10e1c849e8b20c2a693893cdc32025-08-20T03:55:23ZengSpringerSaudi Pharmaceutical Journal1319-01642020-05-0128555055910.1016/j.jsps.2020.03.006Bioassay-guided isolation of anti-hepatitis B virus flavonoid myricetin-3-O-rhamnoside along with quercetin from Guiera senegalensis leavesMohammad K. Parvez0Mohammed S. Al-Dosari1Ahmed H. Arbab2Adnan J. Al-Rehaily3Mazin A.S. Abdelwahid4Department of Pharmacognosy, College of Pharmacy, King Saud University, Riyadh, Saudi Arabia; Corresponding authors at: Department of Pharmacognosy, College of Pharmacy, King Saud University, Riyadh 11451, Saudi Arabia.Department of Pharmacognosy, College of Pharmacy, King Saud University, Riyadh, Saudi Arabia; Corresponding authors at: Department of Pharmacognosy, College of Pharmacy, King Saud University, Riyadh 11451, Saudi Arabia.Department of Pharmacognosy, College of Pharmacy, King Saud University, Riyadh, Saudi Arabia; Department of Pharmacognosy, Faculty of Pharmacy, University of Khartoum, Khartoum, SudanDepartment of Pharmacognosy, College of Pharmacy, King Saud University, Riyadh, Saudi ArabiaDepartment of Pharmaceutical Chemistry, Al-Neelain University, Khartoum, SudanRecently, we have shown in vitro anti-hepatitis B virus (HBV) activity of G. senegalensis J.F. Gmel leaves, and Identified quercetin and other flavonoids by HPTLC. Here we report bioassay-directed fractionation of G. senegalensis leaves using column chromatography and isolation of two flavonoinds from the n-butanol fraction, their structure determination (1H NMR, 13C NMR and 2D-NMR) and assessment of antiviral activities (HBsAg and HBeAg assay) in HBV-reporter HepG2.2.2.15 cells. Further molecular docking was performed against HBV polymerase (Pol/RT) and capsid (Core) proteins as well as host-receptor sodium taurocholate co-transporting polypeptide (NTCP). The two isolated bioactive compounds were identified as quercetin and myricetin-3-O-rhamnoside. Quercetin significantly inhibited synthesis of HBsAg and HBeAg by about 60% and 62%, respectively as compared to myricetin-3-O-rhamnoside by 44% and 35%, respectively. Molecular docking of the two anti-HBV flavonoids revealed their higher binding affinities towards Pol/RT than Core and NTCP. In conclusion, this is the first report on anti-HBV active myricetin-3-O-rhamnoside along with quercetin isolated from G. senegalensis leaves. Their possible mode of anti-HBV activities are suggested through binding with viral Pol/RT and Core as well as host NTCP proteins.http://www.sciencedirect.com/science/article/pii/S131901642030061XGuiera senegalensisMyricetin-3-O-rhamnosideQuercetinHepatitis B virusanti-HBV
spellingShingle Mohammad K. Parvez
Mohammed S. Al-Dosari
Ahmed H. Arbab
Adnan J. Al-Rehaily
Mazin A.S. Abdelwahid
Bioassay-guided isolation of anti-hepatitis B virus flavonoid myricetin-3-O-rhamnoside along with quercetin from Guiera senegalensis leaves
Saudi Pharmaceutical Journal
Guiera senegalensis
Myricetin-3-O-rhamnoside
Quercetin
Hepatitis B virus
anti-HBV
title Bioassay-guided isolation of anti-hepatitis B virus flavonoid myricetin-3-O-rhamnoside along with quercetin from Guiera senegalensis leaves
title_full Bioassay-guided isolation of anti-hepatitis B virus flavonoid myricetin-3-O-rhamnoside along with quercetin from Guiera senegalensis leaves
title_fullStr Bioassay-guided isolation of anti-hepatitis B virus flavonoid myricetin-3-O-rhamnoside along with quercetin from Guiera senegalensis leaves
title_full_unstemmed Bioassay-guided isolation of anti-hepatitis B virus flavonoid myricetin-3-O-rhamnoside along with quercetin from Guiera senegalensis leaves
title_short Bioassay-guided isolation of anti-hepatitis B virus flavonoid myricetin-3-O-rhamnoside along with quercetin from Guiera senegalensis leaves
title_sort bioassay guided isolation of anti hepatitis b virus flavonoid myricetin 3 o rhamnoside along with quercetin from guiera senegalensis leaves
topic Guiera senegalensis
Myricetin-3-O-rhamnoside
Quercetin
Hepatitis B virus
anti-HBV
url http://www.sciencedirect.com/science/article/pii/S131901642030061X
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