Structural Determinants of Oxantel Analogs Reveal Modulatory Selectivity of α3β2 and α4β2 Neuronal Nicotinic Acetylcholine Receptors

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Main Authors: Francesco Bavo, Lucy Chechik, Khoa Huynh, Anna Kolanowski, Avery Richardson, Sydney Tardrew, Nipun Basrur, Mark M. Levandoski, Bente Fro̷lund
Format: Article
Language:English
Published: American Chemical Society 2025-02-01
Series:ACS Omega
Online Access:https://doi.org/10.1021/acsomega.4c11196
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author Francesco Bavo
Lucy Chechik
Khoa Huynh
Anna Kolanowski
Avery Richardson
Sydney Tardrew
Nipun Basrur
Mark M. Levandoski
Bente Fro̷lund
author_facet Francesco Bavo
Lucy Chechik
Khoa Huynh
Anna Kolanowski
Avery Richardson
Sydney Tardrew
Nipun Basrur
Mark M. Levandoski
Bente Fro̷lund
author_sort Francesco Bavo
collection DOAJ
format Article
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institution DOAJ
issn 2470-1343
language English
publishDate 2025-02-01
publisher American Chemical Society
record_format Article
series ACS Omega
spelling doaj-art-061fce3eb7704eebb3b6ec8e2a48437c2025-08-20T03:11:04ZengAmerican Chemical SocietyACS Omega2470-13432025-02-011077338734910.1021/acsomega.4c11196Structural Determinants of Oxantel Analogs Reveal Modulatory Selectivity of α3β2 and α4β2 Neuronal Nicotinic Acetylcholine ReceptorsFrancesco Bavo0Lucy Chechik1Khoa Huynh2Anna Kolanowski3Avery Richardson4Sydney Tardrew5Nipun Basrur6Mark M. Levandoski7Bente Fro̷lund8Department of Drug Design and Pharmacology, University of Copenhagen, Copenhagen, DenmarkDepartment of Chemistry, Program of Neuroscience, Grinnell College, Grinnell, Iowa, United StatesDepartment of Drug Design and Pharmacology, University of Copenhagen, Copenhagen, DenmarkDepartment of Chemistry, Program of Neuroscience, Grinnell College, Grinnell, Iowa, United StatesDepartment of Chemistry, Program of Neuroscience, Grinnell College, Grinnell, Iowa, United StatesDepartment of Chemistry, Program of Neuroscience, Grinnell College, Grinnell, Iowa, United StatesDepartment of Chemistry, Program of Neuroscience, Grinnell College, Grinnell, Iowa, United StatesDepartment of Chemistry, Program of Neuroscience, Grinnell College, Grinnell, Iowa, United StatesDepartment of Drug Design and Pharmacology, University of Copenhagen, Copenhagen, Denmarkhttps://doi.org/10.1021/acsomega.4c11196
spellingShingle Francesco Bavo
Lucy Chechik
Khoa Huynh
Anna Kolanowski
Avery Richardson
Sydney Tardrew
Nipun Basrur
Mark M. Levandoski
Bente Fro̷lund
Structural Determinants of Oxantel Analogs Reveal Modulatory Selectivity of α3β2 and α4β2 Neuronal Nicotinic Acetylcholine Receptors
ACS Omega
title Structural Determinants of Oxantel Analogs Reveal Modulatory Selectivity of α3β2 and α4β2 Neuronal Nicotinic Acetylcholine Receptors
title_full Structural Determinants of Oxantel Analogs Reveal Modulatory Selectivity of α3β2 and α4β2 Neuronal Nicotinic Acetylcholine Receptors
title_fullStr Structural Determinants of Oxantel Analogs Reveal Modulatory Selectivity of α3β2 and α4β2 Neuronal Nicotinic Acetylcholine Receptors
title_full_unstemmed Structural Determinants of Oxantel Analogs Reveal Modulatory Selectivity of α3β2 and α4β2 Neuronal Nicotinic Acetylcholine Receptors
title_short Structural Determinants of Oxantel Analogs Reveal Modulatory Selectivity of α3β2 and α4β2 Neuronal Nicotinic Acetylcholine Receptors
title_sort structural determinants of oxantel analogs reveal modulatory selectivity of α3β2 and α4β2 neuronal nicotinic acetylcholine receptors
url https://doi.org/10.1021/acsomega.4c11196
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