Synthesis, Characterization and Antimicrobial activity Study Via some new Schiff bases for Trimethoprim

This search reports the synthesis of some new series of Schiff base compounds for trimetheprim derivatives which known high been known as a medicinal effectiveness. Trimetheprim was condensed with several substituted aldehydes compounds.(4-dimethyl amine benzaldehyde , propanal , salicaldehyde, 2.4...

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Main Author: Baghdad Science Journal
Format: Article
Language:English
Published: University of Baghdad, College of Science for Women 2010-03-01
Series:مجلة بغداد للعلوم
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Online Access:http://bsj.uobaghdad.edu.iq/index.php/BSJ/article/view/2905
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author Baghdad Science Journal
author_facet Baghdad Science Journal
author_sort Baghdad Science Journal
collection DOAJ
description This search reports the synthesis of some new series of Schiff base compounds for trimetheprim derivatives which known high been known as a medicinal effectiveness. Trimetheprim was condensed with several substituted aldehydes compounds.(4-dimethyl amine benzaldehyde , propanal , salicaldehyde, 2.4 dimethoxy benzaldehyde and 4- methyl benzaldehyde) to obtain Schiff base products(1a-5a) and several substituted ketones compound (4-aminoacetophenone,4-chloroacetophenone, isobutyleketone, acetylacetone and acetophenone) to obtain Schiff base products(6b-10b) in ethanol in the presence of concentrated sulphuric acid as a catalyst to yield the Schiff base. The structure of synthesized compounds has been established on the basis of their Chemical structures of all products were confirmed by spectrophotometric methods such as U.V. visible and FTIR.. All these compounds were evaluated for their antibacterial activity in vitro against Gram + ve bacteria (bacillus) , Gram –ve bacteria (E-Coli).Most Compound under investigation exhibited potent antibacterial activity
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institution Kabale University
issn 2078-8665
2411-7986
language English
publishDate 2010-03-01
publisher University of Baghdad, College of Science for Women
record_format Article
series مجلة بغداد للعلوم
spelling doaj-art-0398e6bfbd0a453b9f5e90ab0d4a85222025-08-20T03:58:10ZengUniversity of Baghdad, College of Science for Womenمجلة بغداد للعلوم2078-86652411-79862010-03-017110.21123/bsj.7.1.614-620Synthesis, Characterization and Antimicrobial activity Study Via some new Schiff bases for TrimethoprimBaghdad Science JournalThis search reports the synthesis of some new series of Schiff base compounds for trimetheprim derivatives which known high been known as a medicinal effectiveness. Trimetheprim was condensed with several substituted aldehydes compounds.(4-dimethyl amine benzaldehyde , propanal , salicaldehyde, 2.4 dimethoxy benzaldehyde and 4- methyl benzaldehyde) to obtain Schiff base products(1a-5a) and several substituted ketones compound (4-aminoacetophenone,4-chloroacetophenone, isobutyleketone, acetylacetone and acetophenone) to obtain Schiff base products(6b-10b) in ethanol in the presence of concentrated sulphuric acid as a catalyst to yield the Schiff base. The structure of synthesized compounds has been established on the basis of their Chemical structures of all products were confirmed by spectrophotometric methods such as U.V. visible and FTIR.. All these compounds were evaluated for their antibacterial activity in vitro against Gram + ve bacteria (bacillus) , Gram –ve bacteria (E-Coli).Most Compound under investigation exhibited potent antibacterial activityhttp://bsj.uobaghdad.edu.iq/index.php/BSJ/article/view/2905"Ttrimetheprim , Schiff bases , aldehyde .ketone, antibacterial activity."
spellingShingle Baghdad Science Journal
Synthesis, Characterization and Antimicrobial activity Study Via some new Schiff bases for Trimethoprim
مجلة بغداد للعلوم
"Ttrimetheprim , Schiff bases , aldehyde .ketone, antibacterial activity."
title Synthesis, Characterization and Antimicrobial activity Study Via some new Schiff bases for Trimethoprim
title_full Synthesis, Characterization and Antimicrobial activity Study Via some new Schiff bases for Trimethoprim
title_fullStr Synthesis, Characterization and Antimicrobial activity Study Via some new Schiff bases for Trimethoprim
title_full_unstemmed Synthesis, Characterization and Antimicrobial activity Study Via some new Schiff bases for Trimethoprim
title_short Synthesis, Characterization and Antimicrobial activity Study Via some new Schiff bases for Trimethoprim
title_sort synthesis characterization and antimicrobial activity study via some new schiff bases for trimethoprim
topic "Ttrimetheprim , Schiff bases , aldehyde .ketone, antibacterial activity."
url http://bsj.uobaghdad.edu.iq/index.php/BSJ/article/view/2905
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