Adverse event profile of five anti head and neck squamous cell carcinoma drugs: a descriptive analysis from WHO-VigiAccess

BackgroundHead and neck squamous cell carcinoma (HNSCC) remains a significant global health concern, with treatment outcomes for advanced or metastatic stages being suboptimal despite the availability of various targeted therapies and immunotherapies. This study evaluates five FDA-approved anti-HNSC...

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Main Authors: Weimin Gao, Zhigang Xia, Tingfeng Zhou, Youlin Dong
Format: Article
Language:English
Published: Frontiers Media S.A. 2025-06-01
Series:Frontiers in Pharmacology
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Online Access:https://www.frontiersin.org/articles/10.3389/fphar.2025.1602276/full
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author Weimin Gao
Zhigang Xia
Tingfeng Zhou
Youlin Dong
author_facet Weimin Gao
Zhigang Xia
Tingfeng Zhou
Youlin Dong
author_sort Weimin Gao
collection DOAJ
description BackgroundHead and neck squamous cell carcinoma (HNSCC) remains a significant global health concern, with treatment outcomes for advanced or metastatic stages being suboptimal despite the availability of various targeted therapies and immunotherapies. This study evaluates five FDA-approved anti-HNSCC drugs—cetuximab, pembrolizumab, nivolumab, atezolizumab, and durvalumab—focusing on the adverse drug reactions (ADRs) associated with their use as reported in the WHO VigiAccess database.MethodsA retrospective analysis was conducted on ADR reports from the WHO-VigiAccess database, focusing on demographic information (age, gender, and geographical distribution) and ADR classification. The disproportionality analysis was used to identify ADRs through Reporting Odds Ratios (ROR) and Proportional Reporting Ratios (PRR). ADRs were categorized into 27 system organ classes (SOCs) for comparison across the five drugs.ResultsA total of 145,678 ADR reports were analyzed. Cetuximab exhibited the highest incidence of skin and subcutaneous tissue disorders (20.88%), while durvalumab showed elevated respiratory system disorders (18.53%). Pembrolizumab and nivolumab had notable immune-related adverse events, with malignant neoplasm progression reported at 5.56% and 4.23%, respectively. Atezolizumab was primarily associated with blood and lymphatic system disorders (5.51%). Disproportionality analysis revealed significant safety concerns for each drug, such as skin toxicity for cetuximab, respiratory complications for durvalumab, and reproductive system risks for nivolumab.ConclusionThis comparative pharmacovigilance study highlights the diverse safety profiles of the five anti-HNSCC drugs. Clinicians should consider these ADRs when treating patients, especially elderly individuals or those with comorbidities. Personalized monitoring strategies should be developed to minimize risks and optimize therapeutic outcomes for HNSCC patients.
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spelling doaj-art-001d81eaa2c74c0887baefa828edc7e82025-08-20T03:29:27ZengFrontiers Media S.A.Frontiers in Pharmacology1663-98122025-06-011610.3389/fphar.2025.16022761602276Adverse event profile of five anti head and neck squamous cell carcinoma drugs: a descriptive analysis from WHO-VigiAccessWeimin Gao0Zhigang Xia1Tingfeng Zhou2Youlin Dong3Department of Otolaryngology, The Second Affiliated Hospital of Jiaxing University, Jiaxing, ChinaDepartment of Otolaryngology, The Second Affiliated Hospital of Jiaxing University, Jiaxing, ChinaDepartment of Otolaryngology, The First Affiliated Hospital of Wenzhou Medical University, Wenzhou, ChinaDepartment of Otolaryngology, The Second Affiliated Hospital of Jiaxing University, Jiaxing, ChinaBackgroundHead and neck squamous cell carcinoma (HNSCC) remains a significant global health concern, with treatment outcomes for advanced or metastatic stages being suboptimal despite the availability of various targeted therapies and immunotherapies. This study evaluates five FDA-approved anti-HNSCC drugs—cetuximab, pembrolizumab, nivolumab, atezolizumab, and durvalumab—focusing on the adverse drug reactions (ADRs) associated with their use as reported in the WHO VigiAccess database.MethodsA retrospective analysis was conducted on ADR reports from the WHO-VigiAccess database, focusing on demographic information (age, gender, and geographical distribution) and ADR classification. The disproportionality analysis was used to identify ADRs through Reporting Odds Ratios (ROR) and Proportional Reporting Ratios (PRR). ADRs were categorized into 27 system organ classes (SOCs) for comparison across the five drugs.ResultsA total of 145,678 ADR reports were analyzed. Cetuximab exhibited the highest incidence of skin and subcutaneous tissue disorders (20.88%), while durvalumab showed elevated respiratory system disorders (18.53%). Pembrolizumab and nivolumab had notable immune-related adverse events, with malignant neoplasm progression reported at 5.56% and 4.23%, respectively. Atezolizumab was primarily associated with blood and lymphatic system disorders (5.51%). Disproportionality analysis revealed significant safety concerns for each drug, such as skin toxicity for cetuximab, respiratory complications for durvalumab, and reproductive system risks for nivolumab.ConclusionThis comparative pharmacovigilance study highlights the diverse safety profiles of the five anti-HNSCC drugs. Clinicians should consider these ADRs when treating patients, especially elderly individuals or those with comorbidities. Personalized monitoring strategies should be developed to minimize risks and optimize therapeutic outcomes for HNSCC patients.https://www.frontiersin.org/articles/10.3389/fphar.2025.1602276/fullHNSCCWHO-vigiaccessanti-HNSCC drugsadverse drug reactionsdisproportionality analysis
spellingShingle Weimin Gao
Zhigang Xia
Tingfeng Zhou
Youlin Dong
Adverse event profile of five anti head and neck squamous cell carcinoma drugs: a descriptive analysis from WHO-VigiAccess
Frontiers in Pharmacology
HNSCC
WHO-vigiaccess
anti-HNSCC drugs
adverse drug reactions
disproportionality analysis
title Adverse event profile of five anti head and neck squamous cell carcinoma drugs: a descriptive analysis from WHO-VigiAccess
title_full Adverse event profile of five anti head and neck squamous cell carcinoma drugs: a descriptive analysis from WHO-VigiAccess
title_fullStr Adverse event profile of five anti head and neck squamous cell carcinoma drugs: a descriptive analysis from WHO-VigiAccess
title_full_unstemmed Adverse event profile of five anti head and neck squamous cell carcinoma drugs: a descriptive analysis from WHO-VigiAccess
title_short Adverse event profile of five anti head and neck squamous cell carcinoma drugs: a descriptive analysis from WHO-VigiAccess
title_sort adverse event profile of five anti head and neck squamous cell carcinoma drugs a descriptive analysis from who vigiaccess
topic HNSCC
WHO-vigiaccess
anti-HNSCC drugs
adverse drug reactions
disproportionality analysis
url https://www.frontiersin.org/articles/10.3389/fphar.2025.1602276/full
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