The GPCR antagonist PPTN synergizes with caspofungin providing increased fungicidal activity against Aspergillus fumigatus by Thaila Fernanda dos Reis, Endrews Delbaje, Camila Figueiredo Pinzan, Rafael Bastos, Suzanne Ackloo, Sara Fallah, Bradley Laflamme, Nicole Robbins, Leah E. Cowen, Gustavo H. Goldman

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Potent and selective SETDB1 covalent negative allosteric modulator reduces methyltransferase activity in cells by Mélanie Uguen, Devan J. Shell, Madhushika Silva, Yu Deng, Fengling Li, Magdalena M. Szewczyk, Ka Yang, Yani Zhao, Michael A. Stashko, Jacqueline L. Norris-Drouin, Jarod M. Waybright, Serap Beldar, Justin M. Rectenwald, Angie L. Mordant, Thomas S. Webb, Laura E. Herring, Cheryl H. Arrowsmith, Suzanne Ackloo, Steven P. Gygi, Robert K. McGinty, Dalia Barsyte-Lovejoy, Pengda Liu, Levon Halabelian, Lindsey I. James, Kenneth H. Pearce, Stephen V. Frye

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OICR-41103 as a chemical probe for the DCAF1 WD40 domain by Serah W. Kimani, Mahmoud Noureldin, Brian Wilson, Laurent Hoffer, Stuart R. Green, Magdalena M. Szewczyk, Héctor González-Álvarez, Mohammed Mohammed, Manuel Chan, Chiara Krausser, Alice Shi Ming Li, Taraneh Hajian, Sarah Tucker, Dhananjay Joshi, Punit Saraon, Brigitte Thériault, Ji Sup Kim, Vijayaratnam Santhakumar, Peter Loppnau, Yanjun Li, Almagul Seitova, Aiping Dong, Taira Kiyota, Tobias Hammann, Paul Gehrtz, Bhashant Patel, Vaibhavi Rathod, Anand Vala, Bhimsen Rout, Paras Jagodra, Peter J. Brown, Ahmed Aman, Jailall Ramnauth, Gennady Poda, David Uehling, Cheryl H. Arrowsmith, Dalia Barsyte-Lovejoy, Richard Marcellus, Suzanne Ackloo, Ahmed Mamai, Rima Al-awar, Levon Halabelian

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Crystal structures of DCAF1-PROTAC-WDR5 ternary complexes provide insight into DCAF1 substrate specificity by Mark F. Mabanglo, Brian Wilson, Mahmoud Noureldin, Serah W. Kimani, Ahmed Mamai, Chiara Krausser, Héctor González-Álvarez, Smriti Srivastava, Mohammed Mohammed, Laurent Hoffer, Manuel Chan, Jamie Avrumutsoae, Alice Shi Ming Li, Taraneh Hajian, Sarah Tucker, Stuart Green, Magdalena Szewczyk, Dalia Barsyte-Lovejoy, Vijayaratnam Santhakumar, Suzanne Ackloo, Peter Loppnau, Yanjun Li, Almagul Seitova, Taira Kiyota, Jue George Wang, Gilbert G. Privé, Douglas A. Kuntz, Bhashant Patel, Vaibhavi Rathod, Anand Vala, Bhimsen Rout, Ahmed Aman, Gennady Poda, David Uehling, Jailall Ramnauth, Levon Halabelian, Richard Marcellus, Rima Al-awar, Masoud Vedadi

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