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Design, Synthesis and Pharmacological Characterization of the First Photoswitchable Small-Molecule Agonist for the Atypical Chemokine Receptor 3 by Sophie Bérenger, Justyna M. Adamska, Francesca Deflorian, Chris de Graaf, Christie B. Palmer, Martyna Szpakowska, Andy Chevigné, Iwan J. P. de Esch, Barbara Zarzycka, Henry F. Vischer, Maikel Wijtmans, Rob Leurs
Published 2025-02-01Get full text
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Structural visualization of small molecule recognition by CXCR3 uncovers dual-agonism in the CXCR3-CXCR7 system by Shirsha Saha, Fumiya K. Sano, Saloni Sharma, Manisankar Ganguly, Annu Dalal, Sudha Mishra, Divyanshu Tiwari, Hiroaki Akasaka, Takaaki A. Kobayashi, Nabarun Roy, Nashrah Zaidi, Yuzuru Itoh, Rob Leurs, Ramanuj Banerjee, Wataru Shihoya, Osamu Nureki, Arun K. Shukla
Published 2025-03-01Get full text
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