Diverse modes of galacto-specific carbohydrate recognition by a family 31 glycoside hydrolase from Clostridium perfringens. by Julie M Grondin, Da Duan, Alyssa C Kirlin, Kento T Abe, Seth Chitayat, Holly L Spencer, Craig Spencer, Alisha Campigotto, Scott Houliston, Cheryl H Arrowsmith, John S Allingham, Alisdair B Boraston, Steven P Smith

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Structural basis of TMPRSS11D specificity and autocleavage activation by Bryan J. Fraser, Ryan P. Wilson, Sára Ferková, Olzhas Ilyassov, Jackie Lac, Aiping Dong, Yen-Yen Li, Alma Seitova, Yanjun Li, Zahra Hejazi, Tristan M. G. Kenney, Linda Z. Penn, Aled Edwards, Richard Leduc, Pierre-Luc Boudreault, Gregg B. Morin, François Bénard, Cheryl H. Arrowsmith

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PRMT1 inhibitor MS023 suppresses RNA splicing to sensitize small cell lung cancer to DNA damaging agents by Mansi K. Aparnathi, Sami Ul Haq, Jonathan St-Germain, Kevin C.J. Nixon, Joseph Walton, Lifang Song, Safa Majeed, Parasvi S. Patel, Ratheesh Subramaniam, Vivek Philip, Richard Marcellus, Dalia Barsyte-Lovejoy, Rima Al-Awar, Razqallah Hakem, Cheryl H. Arrowsmith, Laurie Ailles, Brian Raught, Benjamin H. Lok

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Potent and selective SETDB1 covalent negative allosteric modulator reduces methyltransferase activity in cells by Mélanie Uguen, Devan J. Shell, Madhushika Silva, Yu Deng, Fengling Li, Magdalena M. Szewczyk, Ka Yang, Yani Zhao, Michael A. Stashko, Jacqueline L. Norris-Drouin, Jarod M. Waybright, Serap Beldar, Justin M. Rectenwald, Angie L. Mordant, Thomas S. Webb, Laura E. Herring, Cheryl H. Arrowsmith, Suzanne Ackloo, Steven P. Gygi, Robert K. McGinty, Dalia Barsyte-Lovejoy, Pengda Liu, Levon Halabelian, Lindsey I. James, Kenneth H. Pearce, Stephen V. Frye

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OICR-41103 as a chemical probe for the DCAF1 WD40 domain by Serah W. Kimani, Mahmoud Noureldin, Brian Wilson, Laurent Hoffer, Stuart R. Green, Magdalena M. Szewczyk, Héctor González-Álvarez, Mohammed Mohammed, Manuel Chan, Chiara Krausser, Alice Shi Ming Li, Taraneh Hajian, Sarah Tucker, Dhananjay Joshi, Punit Saraon, Brigitte Thériault, Ji Sup Kim, Vijayaratnam Santhakumar, Peter Loppnau, Yanjun Li, Almagul Seitova, Aiping Dong, Taira Kiyota, Tobias Hammann, Paul Gehrtz, Bhashant Patel, Vaibhavi Rathod, Anand Vala, Bhimsen Rout, Paras Jagodra, Peter J. Brown, Ahmed Aman, Jailall Ramnauth, Gennady Poda, David Uehling, Cheryl H. Arrowsmith, Dalia Barsyte-Lovejoy, Richard Marcellus, Suzanne Ackloo, Ahmed Mamai, Rima Al-awar, Levon Halabelian

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