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Multiple intramolecular triggers converge to preferential G protein coupling in the CB2R by Adrian Morales-Pastor, Tamara Miljuš, Miguel Dieguez-Eceolaza, Tomasz Maciej Stępniewski, Vicente Ledesma-Martin, Franziska M. Heydenreich, Tilman Flock, Bianca Plouffe, Christian Le Gouill, Jean Duchaine, David A. Sykes, Colin Nicholson, Eline J. Koers, Wolfgang Guba, Arne C. Rufer, Uwe Grether, Michel Bouvier, Dmitry B. Veprintsev, Jana Selent
Published 2025-06-01Get full text
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A universal cannabinoid CB1 and CB2 receptor TR-FRET kinetic ligand-binding assay by Leire Borrega-Roman, Leire Borrega-Roman, Leire Borrega-Roman, Leire Borrega-Roman, Bradley L. Hoare, Bradley L. Hoare, Miroslav Kosar, Roman C. Sarott, Kacper J. Patej, Jara Bouma, Morgan Scott-Dennis, Morgan Scott-Dennis, Eline J. Koers, Eline J. Koers, Thais Gazzi, Leonard Mach, Sergio Barrondo, Sergio Barrondo, Sergio Barrondo, Joan Sallés, Joan Sallés, Joan Sallés, Wolfgang Guba, Eric Kusznir, Marc Nazaré, Arne C. Rufer, Uwe Grether, Laura H. Heitman, Erick M. Carreira, David A. Sykes, David A. Sykes, Dmitry B. Veprintsev, Dmitry B. Veprintsev
Published 2025-04-01Get full text
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Enhancing Drug Discovery and Development through the Integration of Medicinal Chemistry, Chemical Biology, and Academia-Industry Partnerships: Insights from Roche’s Endocannabinoid... by Johannes Aebi, Kenneth Atz, Simon M. Ametamey, Jörg Benz, Julie Blaising, Stefania Butini, Giuseppe Campiani, Erick M. Carreira, Ludovic Collin, Eva de Lago, Thais Gazzi, Jürg Gertsch, Luca Gobbi, Wolfgang Guba, Javier Fernández-Ruiz, Jürgen Fingerle, Achi Haider, Yingfang He, Laura H. Heitman, Michael Honer, Daniel Hunziker, Bernd Kuhn, Mauro Maccarrone, Hans Peter Märki, Rainer E. Martin, Peter Mohr, Linjing Mu, Marc Nazaré, David F. Nippa, Sergio Oddi, Fionn O’Hara, Pal Pacher, Julian Romero, Stephan Röver, Arne C. Rufer, Roger Schibli, Gisbert Schneider, Antonia F. Stepan, David A. Sykes, Christoph Ullmer, Mario van der Stelt, Dmitry B. Veprintsev, Matthias B. Wittwer, Uwe Grether
Published 2024-08-01Get full text
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